Formulations for PK/Efficacy/Tox Studies
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Ongoing, First published Apr 08, 2024
https://www.crystalpharmatech.com/preclinical-formulation-development/


Preclinical Formulation for PK/Efficacy/Tox Studies
Contrary to popular belief, early preclinical formulation development is not simply dumping API in a vehicle and gavage feeding an animal. If you do this, you will most likely lose time and money with unnecessary and confusing PK studies. This led to the development of our SMART biopharmaceutical solutions that offer input from our scientific advisory board: A one-stop shop from candidate selection through GMP FIH.
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πš‚πš™πš˜πš’πš•πšŽπš›πšœ πšπš˜πš› π™Ύπš–πš—πš’πšœπšŒπš’πšŽπš—πš πšπšŽπšŠπšπšŽπš›'𝚜 πš…πš’πšŽπš πš™πš˜πš’πš—πš πšŠπš‘πšŽπšŠπš! πš†πš‘πšŽπš›πšŽπš’πš—: 𝙰 πšπš’πš›πš•, πšœπš™πš˜πš’πš•πšŽπš 𝚊𝚜 πšŒπšŠπš— πš‹πšŽ, πš›πšŽπšŠπš•πš’πš£πšŽπšœ πšπš‘πšŠπš πšœπš‘πšŽ πšŒπšŠπš—'𝚝 πšπš•πšŠπšžπš—πš πšπšŠπšπš‘πšŽπš›'𝚜 πšŒπš˜πš–πš™πšŠπš—πš’ πš’πš— 𝚊 πš πš˜πš›πš•πš πšπš˜πš–πš’πš—πšŠπšπšŽπš πš‹πš’ πšπš‘πšŽ πš‚π™²π™΄π™½π™°πšπ™Έπ™Ύ. πšƒπš˜πšœπšœπš’πš—πš πšŠπšœπš’πšπšŽ πš™πšŽπšπšπš’ πšŒπš˜πš›πš™πš˜πš›πšŠπšπš’πš˜πš—πšœ πšŠπš—πš πšŽπš—πšπšŽπš›πš™πš›πš’πšœπšŽπšœ, πšœπš‘πšŽ 𝚜𝚎𝚝𝚜 πš‘πšŽπš› πš•πš˜πšπšπš’ πšœπš’πšπš‘πšπšœ πš‘πšŽπšŠπšŸπšŽπš—πš πšŠπš›πš; πšŠπš’πš–πš’πš—πš 𝚝𝚘 πšπš’πš—πš 𝚊 𝚠𝚊𝚒 𝚝𝚘 πšŽπš‘πš™πš•πš˜πš’πš πšπš‘πšŽ πš‚πšƒπ™°πš πš‚πšƒπšπ™΄π™°π™Ό πš’πšπšœπšŽπš•πš.
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πš‚πš™πš˜πš’πš•πšŽπš›πšœ πšπš˜πš› π™Ύπš–πš—πš’πšœπšŒπš’πšŽπš—πš πšπšŽπšŠπšπšŽπš›'𝚜 πš…πš’πšŽπš πš™πš˜πš’πš—πš πšŠπš‘πšŽπšŠπš! πš†πš‘πšŽπš›πšŽπš’πš—: 𝙰 πšπš’πš›πš•, πšœπš™πš˜πš’πš•πšŽπš 𝚊𝚜 πšŒπšŠπš— πš‹πšŽ, πš›πšŽπšŠπš•πš’πš£πšŽπšœ πšπš‘πšŠπš πšœπš‘πšŽ πšŒπšŠπš—'𝚝 πšπš•πšŠπšžπš—πš πšπšŠπšπš‘πšŽπš›'𝚜 πšŒπš˜πš–πš™πšŠπš—πš’ πš’πš— 𝚊 πš πš˜πš›πš•πš πšπš˜πš–πš’πš—πšŠπšπšŽπš πš‹πš’ πšπš‘πšŽ πš‚π™²π™΄π™½π™°πšπ™Έπ™Ύ. πšƒπš˜πšœπšœπš’πš—πš πšŠπšœπš’πšπšŽ πš™πšŽπšπšπš’ πšŒπš˜πš›πš™πš˜πš›πšŠπšπš’πš˜πš—πšœ πšŠπš—πš πšŽπš—πšπšŽπš›πš™πš›πš’πšœπšŽπšœ, πšœπš‘πšŽ 𝚜𝚎𝚝𝚜 πš‘πšŽπš› πš•πš˜πšπšπš’ πšœπš’πšπš‘πšπšœ πš‘πšŽπšŠπšŸπšŽπš—πš πšŠπš›πš; πšŠπš’πš–πš’πš—πš 𝚝𝚘 πšπš’πš—πš 𝚊 𝚠𝚊𝚒 𝚝𝚘 πšŽπš‘πš™πš•πš˜πš’πš πšπš‘πšŽ πš‚πšƒπ™°πš πš‚πšƒπšπ™΄π™°π™Ό πš’πšπšœπšŽπš•πš.